Azelaic acid is a naturally occurring dicarboxylic acid found in whole grain cereals, rye, and barley and animal products. It is FDA approved as a topical preparation for treatment of acne and is effective against a number of other skin conditions when applied topically. There is strong scientific evidence that Azelaic Acid and Zinc are potent inhibitors of 5-Alpha-Reductase. When Azelaic acid, Vitamin B6 and Zinc Sulfate where added together at very low concentrations, 90% inhibition of 5 Alpha-Reductase activity was obtained. The synergistic activity of these compounds against 5-Alpha-Reductase makes this combination very effective in treatment of male pattern baldness.

By combining GLA, ALA, Linoleic Acid, Azelaic acid, Vitamin B6, Zinc Sulfate and Saw Palmetto extract, we have created a natural yet extremely powerful anti-DHT formula. These ingredients work through different mechanisms to synergistically inhibit both type 1 and 2 forms of 5-Alpha Reductase and decrease DHT locally. By decreasing the DHT levels, hair follicles can grow and thicken naturally, leading to a fuller, healthier scalp without the side effects associated with synthetic drugs.

Saw palmetto has been extensively studied over the past several years for the treatment of enlarged prostate in men ( BPH ). Saw Palmetto extract which is a known anti-androgen is the liposerolic extract of the fruit of Saw Palmetto.

Saw Palmetto has shown to effectively block DHT and is also believed to block the androgen receptors which are found on the hair follicles. Like GLA and ALA it also blocks Type 1 and Type 2 forms of 5 alpha-reductase and has shown to be more potent than Finasteride, the active ingredient of Propecia.